Tacrolimus

Product: Urolithin A

Identifier : DBSNPE000126
Drug : DB00864 (Tacrolimus)
Interacting Gene/Enzyme : Multidrug resistance protein 1
Gene Name : ABCB1
UniProt ID : P08183
Defining Change(s) :

  • T Allele (G2677T) (rs2032582 )

Allele Name : Not Available
Genotype(s) : (T;T) / (G;T)
Type(s) : ADR Directly Studied
Groups : Not Available
Description : Increased risk of neurotoxicity
References :

  1. Yamauchi A, Ieiri I, Kataoka Y, Tanabe M, Nishizaki T, Oishi R, Higuchi S, Otsubo K, Sugimachi K: Neurotoxicity induced by tacrolimus after liver divansplantation: relation to genetic polymorphisms of the ABCB1 (MDR1) gene. Transplantation. 2002 Aug 27;74(4):571-2. [PubMed:12352921 ]

PMID: 24358263

Tacrolimus

Product: BAY1217389

Identifier : DBSNPE000243
Drug : DB00864 (Tacrolimus)
Interacting Gene/Enzyme : Cytochrome P450 3A5
Gene Name : CYP3A5
UniProt ID : P20815
Defining Change(s) :

  • Functional gene

Allele Name : CYP3A5*1
Genotype(s) : Not Available
Type(s) : Effect Directly Studied
Groups : Not Available
Description : Higher dose requirement (1.5-2x)
References :

  1. Birdwell KA, Decker B, Barbarino JM, Peterson JF, Stein CM, Sadee W, Wang D, Vinks AA, He Y, Swen JJ, Leeder JS, van Schaik R, Thummel KE, Klein TE, Caudle KE, MacPhee IA: Clinical Pharmacogenetics Implementation Consortium (CPIC) Guidelines for CYP3A5 Genotype and Tacrolimus Dosing. Clin Pharmacol Ther. 2015 Jul;98(1):19-24. doi: 10.1002/cpt.113. Epub 2015 Jun 3. [PubMed:25801146 ]

PMID: 8473300

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