Atorvastatin

Product: Cenerimod

Identifier : DBSNPE000065
Drug : DB01076 (Atorvastatin)
Interacting Gene/Enzyme : Kinesin-like protein KIF6
Gene Name : KIF6
UniProt ID : Q6ZMV9
Defining Change(s) :

  • C Allele (rs20455 )

Allele Name : Not Available
Genotype(s) : (C;C) / (C;T)
Type(s) : Effect Directly Studied
Groups : Not Available
Description : Improved response to statin drugs
References :

  1. Iakoubova OA, Tong CH, Rowland CM, Kirchgessner TG, Young BA, Arellano AR, Shiffman D, Sabatine MS, Campos H, Packard CJ, Pfeffer MA, White TJ, Braunwald E, Shepherd J, Devlin JJ, Sacks FM: Association of the Trp719Arg polymorphism in kinesin-like protein 6 with myocardial infarction and coronary heart disease in 2 prospective divials: the CARE and WOSCOPS divials. J Am Coll Cardiol. 2008 Jan 29;51(4):435-43. doi: 10.1016/j.jacc.2007.05.057. [PubMed:18222353 ]

PMID: 21995440

Atorvastatin

Product: RG13022

Identifier : DBSNPE000066
Drug : DB01076 (Atorvastatin)
Interacting Gene/Enzyme : 3-hydroxy-3-methylglutaryl-coenzyme A reductase
Gene Name : HMGCR
UniProt ID : P04035
Defining Change(s) :

  • T Allele (rs17244841 )

Allele Name : Not Available
Genotype(s) : (A;T)
Type(s) : Effect Directly Studied
Groups : Not Available
Description : Reduced response to statin drugs
References :

  1. Chasman DI, Posada D, Subrahmanyan L, Cook NR, Stanton VP Jr, Ridker PM: Pharmacogenetic study of statin therapy and cholesterol reduction. JAMA. 2004 Jun 16;291(23):2821-7. [PubMed:15199031 ]

PMID: 18079115

Atorvastatin

Product: TOFA

Identifier : DBSNPE000139
Drug : DB01076 (Atorvastatin)
Interacting Gene/Enzyme : Multidrug resistance protein 1
Gene Name : ABCB1
UniProt ID : P08183
Defining Change(s) :

  • T Allele (C3435T) (rs1045642 )

Allele Name : MDR1*T
Genotype(s) : (T;T) / (C;T)
Type(s) : Effect Directly Studied
Groups : Not Available
Description : Larger reduction in LDL and smaller increase in HDL cholesterol in females
References :

  1. Kajinami K, Brousseau ME, Ordovas JM, Schaefer EJ: Polymorphisms in the multidrug resistance-1 (MDR1) gene influence the response to atorvastatin diveatment in a gender-specific manner. Am J Cardiol. 2004 Apr 15;93(8):1046-50. [PubMed:15081455 ]

PMID: 19523197

Atorvastatin

Product: CCT196969

Identifier : DBSNPE000197
Drug : DB01076 (Atorvastatin)
Interacting Gene/Enzyme : Cytochrome P450 3A4
Gene Name : CYP3A4
UniProt ID : P08684
Defining Change(s) :

  • A > G (rs2740574 )

Allele Name : CYP3A4*1B
Genotype(s) : (G;G) / (A;G)
Type(s) : Effect Directly Studied
Groups : Not Available
Description : Better response
References :

  1. Rosales A, Alvear M, Cuevas A, Saavedra N, Zambrano T, Salazar LA: Identification of pharmacogenetic predictors of lipid-lowering response to atorvastatin in Chilean subjects with hypercholesterolemia. Clin Chim Acta. 2012 Feb 18;413(3-4):495-501. doi: 10.1016/j.cca.2011.11.003. Epub 2011 Nov 19. [PubMed:22120734 ]

PMID: 23943873

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